Rearrangement of 3,3-Disubstituted Indolenines and Synthesis of 2,3-Substituted Indoles

200677 citationsJournal Article

Authors

Albert J. Robichaud · Princeton University

Abstract

Synthesis of 2,3-substituted indoles from phenylhydrazine and alpha-branched aldehydes via rearrangement of 3,3-disubstituted indolenine intermediates is reported. [reaction: see text]

Topics & Keywords

Catalytic C–H Functionalization Methods Asymmetric Synthesis and Catalysis Catalytic Cross-Coupling Reactions

Publication Details

Published in: Organic Letters

Volume 8, Issue 25, pp. 5769-5771

DOI: 10.1021/ol0623567

Field-Weighted Citation Impact: 2.86

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Rearrangement of 3,3-Disubstituted Indolenines and Synthesis of 2,3-Substituted Indoles

Authors

Abstract

Topics & Keywords

Publication Details